30 mg CAB (single dose)# [42] |
|
|
|
Cmax (µg/ml) |
3.61 |
3.07 |
1.18 |
AUC0-inf (µg.h/ml) |
146 |
98.2 |
1.49 |
30 mg CAB (repeated doses)# [34] |
|
|
|
Ctrough (µg/ml) |
4.9 |
4.6 |
1.06 |
Cmax (µg/ml) |
8.3 |
7.8 |
1.06 |
AUC0-24 (µg.h/ml) |
147 |
154 |
1.05 |
25 mg RPV (repeated doses)^ [43] |
|
|
|
Cmin (ng/mL) |
89.85 |
68.9 |
1.30 |
Cmax (ng/mL) |
203.8 |
219.75 |
1.08 |
AUC0-24 (ng.h/mL) |
2589 |
3304.9 |
1.28 |
25 mg RPV (repeated doses)^ [45] |
|
|
|
Ctrough (ng/mL) |
67.3 |
62.2 |
1.08 |
Cmax (ng/mL) |
180.9 |
189.60 |
1.05 |
AUC0-24 (ng.h/mL) |
2528 |
2895.7 |
1.15 |
25 mg RPV (repeated doses)# [44] |
|
|
|
Ctrough (ng/mL) |
74.5 |
62.7 |
1.19 |
Cmax (ng/mL) |
148 |
176.01 |
1.19 |
AUC0-24 (ng.h/mL) |
2227 |
2779.8 |
1.25 |
25 mg RPV (repeated doses)# [44] |
|
|
|
Ctrough (ng/mL) |
87.4 |
66.7 |
1.31 |
Cmax (ng/mL) |
171 |
177.68 |
1.04 |
AUC0-24 (ng.h/mL) |
2473 |
2860.3 |
1.16 |
150 mg RPV (repeated doses)^ [46] |
|
|
|
Ctrough (ng/mL) |
478 |
400.6 |
1.19 |
Cmax (ng/mL) |
1123 |
1296 |
1.15 |
AUC0-24 (ng.h/mL) |
16051 |
19398 |
1.21 |
400 mg RAL (repeated doses)# [47] |
|
|
|
Ctrough (ng/ml) |
48.84 |
44.71 |
1.09 |
Cmax (ng/ml) |
1203 |
1749 |
1.45 |
AUC0-12 (ng.h/ml) |
4440 |
8530 |
1.92 |
400 mg RAL (single dose)# [48] |
|
|
|
Ctrough (ng/ml) |
35.79 |
65.65 |
1.83 |
Cmax (ng/ml) |
1279 |
1631 |
1.28 |
AUC0-inf (ng.h/ml) |
4884 |
8406 |
1.72 |