Expressor group (n = 5) Non-expressor group (n = 5)
P-value
Dose (mg) 4 (3-5) 2 (1-3) 0.016
Weight (kg) 54 (51.3-78.0) 65 (43-82) 0.690
Dose/Weight (mg/kg) 0.077 (0.045-0.097) 0.037 (0.016-0.047) 0.032
AUC in Tac BID (ng·hr/mL) 126.3 (98.2-146.9) 107.0 (102.4-126.7) 0.310
AUC in Tac QD (ng·hr/mL) 112.5 (81.0-168.6) 96.1 (68.5-131.7) 0.310
Cmin in Tac BID (mg/mL) 3.77 (3.05-4.20) 3.07 (2.76-4.47) 0.421
Cmin in Tac QD (mg/mL) 3.04 (1.85-4.21) 2.59 (1.81-4.47) 0.690
Cmax in Tac BID (mg/mL) 8.20 (4.94-11.54) 9.93 (5.08-10.48) 0.690
Cmax in Tac QD (mg/mL) 9.52 (6.81-11.90) 7.85 (3.54-10.86) 0.151
Dose-adjusted Cmin in Tac BID (ng/mL/mg) 0.918 (0.754-1.050) 1.535 (0920-3.400) 0.056
Dose-adjusted Cmin in Tac QD (ng/mL/mg) 0.680 (0.608-1.053) 1.295 (0.603-2.235) 0.151
Dose-adjusted Cmax in Tac BID (ng/mL/mg) 1.65 (1.58-2.40) 3.79 (3.31-5.16) 0.008
Dose-adjusted Cmax in Tac QD (ng/mL/mg) 2.73 (1.36-3.10) 3.54 (1.85-5.43) 0.310
Dose-adjusted AUC in Tac BID (ng·hr/mL/mg) 29.4 (25.3-33.0) 53.5 (35.2-102.4) 0.008
Dose-adjusted AUC in Tac QD (ng·hr/mL/mg) 27.0 (21.0-42.2) 48.0 (24.2-68.5) 0.095
Dose/kg-adjusted Cmin Tac BID (ng/mL/mg/kg) 0.015 (0.013-0.018) 0.021 (0.012-0.053) 0.548
Dose/kg-adjusted Cmin Tac QD (ng/mL/mg/kg) 0.013 (0.009-0.014) 0.017 (0.009-0.052) 0.222
Dose/kg-adjusted Cmax Tac BID (ng/mL/mg/kg) 0.032 (0.020-0.046) 0.069 (0.040-0.088) 0.032
Dose/kg-adjusted Cmax Tac QD (ng/mL/mg/kg) 0.038 (0.025-0.052) 0.053 (0.029-0.126) 0.421
Dose/kg-adjusted AUC Tac BID (ng·hr/mL/mg/kg) 0.492 (0.423-0.553) 0.716 (0.455-1.600) 0.151
Dose/kg-adjusted AUC Tac QD (ng·hr/mL/mg/kg) 0.458 (0.390-0.541) 0.643 (0.379-1.532) 0.421